Ipamorelin vs Exenatide

A detailed comparison to help you understand the differences and choose the right peptide for your research goals.

Ipamorelin

Ipamorelin is a selective growth hormone secretagogue that stimulates the release of growth hormone from the pituitary gland without significantly affecting cortisol or prolactin.

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Exenatide

Exenatide was the first GLP-1 receptor agonist approved in the US, derived from a compound found in Gila monster saliva. Available as Byetta (twice daily) and Bydureon (once weekly extended-release).

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Side-by-Side Comparison

AspectIpamorelinExenatide
MechanismActs as a ghrelin mimetic, binding to the ghrelin receptor (GHS-R) in the pituitary to stimulate GH release. Highly selective with minimal effect on other hormones.Synthetic version of exendin-4, which activates GLP-1 receptors to enhance glucose-dependent insulin secretion, suppress glucagon, slow gastric emptying, and promote satiety.
Typical DosageTypical dosing ranges from 200-300mcg administered 2-3 times daily, often combined with CJC-1295.Byetta: 5mcg twice daily for 1 month, then 10mcg twice daily. Bydureon: 2mg subcutaneously once weekly.
AdministrationSubcutaneous injection. Best results when administered fasted or before sleep. Often stacked with GHRH peptides.Byetta: Inject within 60 minutes before morning and evening meals. Bydureon: Any time of day, with or without meals. Do not mix with insulin in same syringe.
Side EffectsGenerally well-tolerated. May cause mild headaches, lightheadedness, or increased hunger initially.Nausea (especially initially), vomiting, diarrhea, dizziness, headache, and injection site reactions (particularly with Bydureon).
Best For

What They Have in Common

Both Ipamorelin and Exenatide are commonly used for:

Key Differences

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